Drug Information

Drug General Information
Drug ID
D02WWM
Former ID
DIB020288
Drug Name
LY97241
Synonyms
LY 97241; LY-97241
Drug Type
Small molecular drug
Indication Discovery agent Investigative [539683]
Formula
C19H32N2O2
InChI
InChI=1S/C19H32N2O2/c1-3-5-6-7-9-16-20(4-2)17-10-8-11-18-12-14-19(15-13-18)21(22)23/h12-15H,3-11,16-17H2,1-2H3
InChIKey
YTYATOMQOOFRNA-UHFFFAOYSA-N
PubChem Compound ID
175064
PubChem Substance ID
7979832, 10258166, 15000076, 25408240, 33499005, 57395179, 77416882, 103450844, 104040005, 104424558, 129847631, 129984347, 135153260, 135650562, 224862993, 232099015
Target and Pathway
Target(s) Kv10.1 Target Info Blocker (channel blocker) [526508]
Kv10.2 Target Info Blocker (channel blocker) [527048]
References
Ref 539683(http://www.guidetopharmacology.org/) Nucleic Acids Res. 2015 Oct 12. pii: gkv1037. The IUPHAR/BPS Guide to PHARMACOLOGY in 2016: towards curated quantitative interactions between 1300 protein targets and 6000 ligands. (Ligand id: 2606).
Ref 526508Inhibition of hEAG1 and hERG1 potassium channels by clofilium and its tertiary analogue LY97241. Br J Pharmacol. 2003 Jan;138(1):161-71.
Ref 527048Molecular determinants for high-affinity block of human EAG potassium channels by antiarrhythmic agents. Mol Pharmacol. 2004 May;65(5):1120-9.

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